Discovery of a novel indole series of EP 1 receptor antagonists by scaffold hopping

A Hall, A Billinton, SH Brown, A Chowdhury…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 18, # 8 p. 2684 - 2690

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Citation Number: 14

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... 2 and 4 As part of an ongoing medicinal chemistry programme we were interested in identifying further novel EP 1 receptor antagonists and profiling their potential for the treatment of inflammatory pain. ...