Design, Biologic Evaluation, and SAR of Novel Pseudo??peptide Incorporating Benzheterocycles as HIV??1 Protease Inhibitors
M He, H Zhang, X Yao, M Eckart…
Index: Chemical Biology and Drug Design, , vol. 76, # 2 p. 174 - 180
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Citation Number: 7
Abstract
... Further design and chemical modifications of these inhibitors utilizing structure-based drug design strategies are currently underway. Acknowledgments. ... Nature Reviews: Molecular Cell Biology;1:40–49. ... 2-hydroxymethyl aziridines of biological interest. Tetra Lett;45:1211–1213. ...
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