A Facile Synthesis of N??Boc??Protected Pyrroles by Cyclodehydration of γ??Amino?螃?, β??enals and??enones

O Paulus, G Alcaraz, M Vaultier

Index: Paulus, Olivier; Alcaraz, Gilles; Vaultier, Michel European Journal of Organic Chemistry, 2002 , # 15 p. 2565 - 2572

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Citation Number: 8

Abstract

Abstract A novel series of N-Boc-substituted and fused pyrroles was prepared by cyclodehydration of readily accessible (E)-γ-(tert-butoxycarbonylamino)-α, β-enals and- enones. Functionalisation of the pyrrole ring was then explored with 2-borylated pyrroles in the Suzuki− Miyaura coupling.(© Wiley-VCH Verlag GmbH, 69451 Weinheim, Germany, 2002)