SAR based design of nicotinamides as a novel class of androgen receptor antagonists for prostate cancer

SH Yang, CH Song, HTM Van, E Park…

Index: Journal of Medicinal Chemistry, , vol. 56, # 8 p. 3414 - 3418

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Citation Number: 15

Abstract

... Journal of Medicinal Chemistry. ... Such DIMN analogues as nicotinamides or terephthalamides (7, 8) were prepared by a similar method which has been recently reported to be favorable for easy isolation of final products with moderate to good chemical yield,(17) and N ...

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