Mild and safer preparative method for nonsymmetrical sulfamides via N-sulfamoyloxazolidinone derivatives: Electronic effects affect the transsulfamoylation reactivity
A Borghese, L Antoine, JP Van Hoeck…
Index: Masui, Toshiaki; Kabaki, Mikio; Watanabe, Hideaki; Kobayashi, Tatsuya; Masui, Yoshiyuki Organic Process Research and Development, 2004 , vol. 8, # 3 p. 408 - 410
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Citation Number: 17
Abstract
... Organic Process Research & Development. ... Chemical Product Research & Development, Lilly ... During the development of a process for the preparation of sulfamide 3 (Scheme 2) via the reaction of the aromatic amine 2 with the i-PrNHSO 2 Cl, 1, we discovered a severe thermal ...
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