One??Pot Synthesis of Camalexins and 3, 3′??Biindoles by the Masuda Borylation–Suzuki Arylation (MBSA) Sequence

BOA Tasch, D Antovic, E Merkul…

Index: Tasch, Boris O. A.; Antovic, Dragutin; Merkul, Eugen; Mueller, Thomas J. J. European Journal of Organic Chemistry, 2013 , # 21 p. 4564 - 4569

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Citation Number: 7

Abstract

Abstract The Masuda borylation/Suzuki arylation (MBSA) sequence starting from N- protected 3-iodoindoles has successfully been extended to the coupling of five-membered heterocycles and indoles in the arylation step, which could not be achieved with previously developed MBSA methods. By this approach the one-pot nature of the method as well as the use of a simple catalyst system has been retained. The applicability of the method has ...