N??[2??Methyl??5??(triazol??1??yl) phenyl] pyrimidin??2??amine as a Scaffold for the Synthesis of Inhibitors of Bcr??Abl

F Arioli, S Borrelli, F Colombo, F Falchi, I Filippi…

Index: ChemMedChem, , vol. 6, # 11 p. 2009 - 2018

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Citation Number: 24

Abstract

... ChemMedChem, 6: 2009–2018. doi: 10.1002/cmdc.201100304. ... Volume: Issue: Page: ... Chemistry. All the compounds were obtained by copper(I)-catalyzed azide–alkyne cycloaddition (CuAAC) according to Sharpless conditions,10 between azides 6 and five different alkynes. ...

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