A new approach to allylamines and pyrrolidines
T Gajda, A Zwierzak
Index: Gajda, Tadeusz; Zwierzak, Andrzej Liebigs Annalen der Chemie, 1986 , # 6 p. 992 - 1002
Full Text: HTML
Citation Number: 2
Abstract
Abstract The 1, 4-adducts 3a–c and 4, readily available from the reaction between diethyl N, N-dichlorophosphoramidate (1) and 1, 3-dienes, were found to be convenient precursors for the efficient synthesis of the δ-chloroallylamine hydrochlorides 5a–d and N-phosphorylated allylamines 6a–c and 7. The three-step transformation of 3a–c affords the cis-3, 4- dibromopyrrolidine hydrochlorides 10a–c. The preparation of the 2, 5-dihydro-1H-pyrrole ...
Related Articles:
[Burdi, Douglas F.; Hunt, Rachel; Fan, Lei; Hu, Tao; Wang, Jun; Guo, Zihong; Huang, Zhiqiang; Wu, Chengde; Hardy, Larry; Detheux, Michel; Orsini, Michael A.; Quinton, Maria S.; Lew, Robert; Spear, Kerry Journal of Medicinal Chemistry, 2010 , vol. 53, # 19 p. 7107 - 7118]
A solid-supported phosphine-free ruthenium alkylidene for olefin metathesis in methanol and water
[Connon, Stephen J; Blechert, Siegfried Bioorganic and medicinal chemistry letters, 2002 , vol. 12, # 14 p. 1873 - 1876]