3-(4-Piperidinyl)-and 3-(8-aza-bicyclo [3.2. 1] oct-3-yl)-2-phenyl-1H-indoles as bioavailable h5-HT 2A antagonists

J Crawforth, S Goodacre, R Maxey, S Bourrain…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 10, # 24 p. 2701 - 2703

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Citation Number: 13

Abstract

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. ... In this letter, we describe the synthesis and receptor binding affinities of compounds where the tryptamine side chain has been constrained within a ring. ...