Process Development of a Scaleable Route to (2 R)-[3-(2-Aminopropyl)-1 H-indol-7-yloxy]-N, N-diethylacetamide: A Key Intermediate for AJ-9677, a Potent and …

H Harada, A Fujii, O Odai, S Kato

Index: Organic Process Research and Development, , vol. 8, # 2 p. 238 - 245

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Citation Number: 6

Abstract

... Organic Process Research & Development. ... Chemistry Research Laboratories, Dainippon ... Herein, we describe the process development of a scaleable synthetic route to the corresponding N,N-diethylacetamide derivative 3 of 2 from 7-benzyloxy-1H-indole (4). Reaction of the ...