Fast DKR of Amines Using Isopropyl 2??Methoxyacetate as Acyl Donor

…, K Hult, ARA Palmans, EW Meijer

Index: Veld, Martijn A. J.; Hult, Karl; Palmans, Anja R. A.; Meijer European Journal of Organic Chemistry, 2007 , # 32 p. 5416 - 5421

Full Text: HTML

Citation Number: 24

Abstract

Abstract The dynamic kinetic resolution (DKR) of various primary amine substrates was performed using a modified version of the Bäckvall system. A single equivalent of isopropyl 2-methoxyacetate was used as acyl donor in combination with p-MeO Shvo complex as the racemization catalyst and Novozym 435 as the acylation catalyst. A reaction temperature of 100 C was employed to ensure a high racemization rate. Adding 2, 4-dimethyl-3-pentanol ...

Related Articles:

Synthesis of heterosubstituted hexaarylbenzenes via asymmetric carbonylative couplings of benzyl halides

[Potter, Robert G.; Hughes, Thomas S. Organic Letters, 2007 , vol. 9, # 7 p. 1187 - 1190]

Synthesis of Acyclic Ketones by Catalytic, Bidirectional Homologation of Formaldehyde with Nonstabilized Diazoalkanes. Application of a Chiral Diazomethyl ( …

[Wommack, Andrew J.; Kingsbury, Jason S. Journal of Organic Chemistry, 2013 , vol. 78, # 21 p. 10573 - 10587]

Hydrogen-bond quenching of photodecarbonylation in the solid state and recovery of reactivity by co-crystallization

[Zhang, Jing; Gembicky, Milan; Messerschmidt, Marc; Coppens, Philip Chemical Communications, 2007 , # 23 p. 2399 - 2401]

The Absorption Spectra of Tetracyclones. IV1, 2

[Coan et al. Journal of the American Chemical Society, 1955 , vol. 77, p. 60,62, 63]

Dakin-west synthesis of β-aryl ketones

[Tran, Khanh-Van; Bickar, David Journal of Organic Chemistry, 2006 , vol. 71, # 17 p. 6640 - 6643]

More Articles...