Tetrahedron Letters

An efficient synthesis of N-benzyl-3-sulfonyl glutarimides. Formal synthesis of the aromatase inhibitor AG-1

MY Chang, BR Chang, HM Tai, NC Chang

Index: Chang, Meng-Yang; Chang, Bo-Rui; Tai, Huo-Mu; Chang, Nein-Chen Tetrahedron Letters, 2000 , vol. 41, # 52 p. 10273 - 10276

Full Text: HTML

Citation Number: 46

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... A formal [3+3] cycloaddition strategy to substituted glutarimides was studied. N-Benzyl α-sulfonylacetamides and various α,β-unsaturated esters were used as starting materials. ... Sequential treatment of chloroacetyl chloride with benzylamine and sodium p-toluenesulfinate furnished α- ...

Related Articles:

Reaction of different α-sulfonyl acetamides with methyl acrylate

[Chang, Meng-Yang; Chen, Shui-Tein; Chang, Nein-Chen Tetrahedron, 2002 , vol. 58, # 25 p. 5075 - 5080]

One-pot facile conversion of Baylis–Hillman adduct into N-alkyl 3-(E)-alkylidene-5-substituted sulfonylpiperidine-2, 6-dione. Formal synthesis of tacamonine

[Chen, Chung-Yi; Chang, Meng-Yang; Hsu, Ru-Ting; Chen, Shui-Tein; Chang, Nein-Chen Tetrahedron Letters, 2003 , vol. 44, # 47 p. 8627 - 8630]

1, 8??Diazabicyclo [5.4. 0] undec??7??ene: A Remarkable Base in the Debromination of 4??or 5??Substituted N??Benzyl α??Bromo?螃窿?p??Toluenesulfonylglutarimide

[Chang, Meng-Yang; Lin, John Yi-Chung; Chen, Shui-Tein; Chang, Nein-Chen Journal of the Chinese Chemical Society, 2002 , vol. 49, # 6 p. 1015 - 1024]

More Articles...