Preparation of N-tert-butoxycarbonylthiourea opens the way to protected 2-aminothiazoles
B Schiavi, A Ahond, C Poupat, P Potier
Index: Schiavi, Bruno; Ahond, Alain; Poupat, Christiane; Potier, Pierre Synthetic Communications, 2002 , vol. 32, # 11 p. 1671 - 1674
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Citation Number: 6
Abstract
The aminothiazole group is a very well known “pharmacophore”. It is, therefore, important to have in hand an easy and high yielding method to prepare it. Iwanowicz et al.1-2 View all references have efficiently prepared N,N-bis-tert-butoxycarbonylthiourea 1 from the sodium salt of ...
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