Synlett

N-Carboalkoxy-2-Nitrobenzenesulfonamides: A Practical Preparation of N-Boc-, N-Alloc-, and N-Cbz-Protected Primary Amines

T Fukuyama, M Cheung, T Kan

Index: Fukuyama, Tohru; Cheung, Mui; Kan, Toshiyuki Synlett, 1999 , # 8 p. 1301 - 1303

Full Text: HTML

Citation Number: 63

Abstract

Abstract: N-Carboalkoxy-2-nitrobenzenesulfonamides, readily prepared by acylation of 2- nitrobenzenesulfonamide (o-NsNH2), can be alkylated by either conventional or Mitsunobu protocols. Since the o-nosyl group can be deprotected under mild conditions, a variety of ...

Related Articles:

Fluorous scavenger for parallel preparation of tertiary sulfonamides leading to secondary amines

[Basle, Emmanuel; Jean, Mickael; Gouault, Nicolas; Renault, Jacques; Uriac, Philippe Tetrahedron Letters, 2007 , vol. 48, # 46 p. 8138 - 8140]

The facile preparation of primary and secondary amines via an improved Fukuyama–Mitsunobu procedure. Application to the synthesis of a lung-targeted gene …

[Guisado, Cristina; Waterhouse, Jodie E.; Price, Wayne S.; Jorgensen, Michael R.; Miller, Andrew D. Organic and Biomolecular Chemistry, 2005 , vol. 3, # 6 p. 1049 - 1057]

More Articles...