A binding mode hypothesis of tiagabine confirms liothyronine effect on γ-aminobutyric acid transporter 1 (GAT1)

A Jurik, B Zdrazil, M Holy, T Stockner…

Index: Vogensen, Stine B.; Jorgensen, Lars; Madsen, Karsten K.; Borkar, Nrupa; Wellendorph, Petrine; Skovgaard-Petersen, Jonas; Schousboe, Arne; White, H. Steve; Krogsgaard-Larsen, Povl; Clausen, Rasmus P. Journal of Medicinal Chemistry, 2013 , vol. 56, # 5 p. 2160 - 2164

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Citation Number: 7

Abstract

... Journal of Medicinal ... University of Vienna, Department of Pharmaceutical Chemistry, Division of Drug Design and Medicinal Chemistry, Althanstraße 14 ... structure of the dDAT and topological information from the literature.(22-24) On the basis of a combination of low B-values and ...