Allene synthesis by an asymmetric Baylis–Hillman style reaction on vinylphosphine oxides
DJ Fox, JA Medlock, R Vosser, S Warren
Index: Fox; Medlock; Vosser; Warren Journal of the Chemical Society. Perkin Transactions 1, 2001 , # 18 p. 2240 - 2249
Full Text: HTML
Citation Number: 21
Abstract
A novel reaction has been discovered with a mechanism similar to the Baylis–Hillman reaction. Reaction of a vinylic phosphine oxide with (R)-N-lithio-α-methylbenzylbenzylamine 2 in the presence of an aldehyde gave hydroxyphosphine oxides in good to moderate yields and moderate to poor enantioselectivities. The hydroxyphosphine oxides undergo the Horner–Wittig elimination reaction to produce allenes. Baylis–Hillman reactions of vinylic ...
Related Articles:
[Takaki, Ken; Takeda, Mitsuhiro; Koshoji, Go; Shishido, Tetsuya; Takehira, Katsuomi Tetrahedron Letters, 2001 , vol. 42, # 36 p. 6357 - 6360]
[Takaki, Ken; Takeda, Mitsuhiro; Koshoji, Go; Shishido, Tetsuya; Takehira, Katsuomi Tetrahedron Letters, 2001 , vol. 42, # 36 p. 6357 - 6360]
[Takaki, Ken; Takeda, Mitsuhiro; Koshoji, Go; Shishido, Tetsuya; Takehira, Katsuomi Tetrahedron Letters, 2001 , vol. 42, # 36 p. 6357 - 6360]
[Davidson,A.H. et al. Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1977 , p. 550 - 565]
[Davidson,A.H. et al. Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1977 , p. 550 - 565]