Novel methods for the synthesis of functionalized indoles from arylhydroxylamines and activated acetylenes
JR Hwu, HV Patel, RJ Lin, MO Gray
Index: Hwu, Jih Ru; Patel, Himatkumar V.; Lin, Ren Jye; Gray, Marissa O. Journal of Organic Chemistry, 1994 , vol. 59, # 6 p. 1577 - 1582
Full Text: HTML
Citation Number: 36
Abstract
Many naturally occurring indoles possess important biological activity.'-'On the other hand, synthetic indoles with substituents at various positions have been used extensively in medicine and pharmacology?* 6* 6 as well as in ho1ography. l Thus, the development of new, efficient method~ l-'*~-~ o that lead to indoles is necessary. Herein, we report two novel methods for the synthesis of indoles which allow easy functionaliiation at almost all ...
Related Articles:
[Melkonyan, Ferdinand S.; Karchava, Alexander V.; Yurovskaya, Marina A. Journal of Organic Chemistry, 2008 , vol. 73, # 11 p. 4275 - 4278]
Ferric chloride-catalyzed synthesis of indoles using the intramolecular amination of aryl bromides
[Melkonyan; Topolyan; Karchava; Yurovskaya Chemistry of Heterocyclic Compounds, 2010 , vol. 46, # 9 p. 1158 - 1160]
[Melkonyan, Ferdinand S.; Karchava, Alexander V.; Yurovskaya, Marina A. Journal of Organic Chemistry, 2008 , vol. 73, # 11 p. 4275 - 4278]
Preparation of spiroindolines as potential intermediates in aspidosperma alkaloid synthesis
[Troin, Yves; Sinibaldi, Marie-Eve; Gramain, Jean-Claude; Rubiralta, Mario; Diez, Anna Tetrahedron Letters, 1991 , vol. 32, # 43 p. 6129 - 6132]
Preparation of spiroindolines as potential intermediates in aspidosperma alkaloid synthesis
[Troin, Yves; Sinibaldi, Marie-Eve; Gramain, Jean-Claude; Rubiralta, Mario; Diez, Anna Tetrahedron Letters, 1991 , vol. 32, # 43 p. 6129 - 6132]