Structure-based design of orally bioavailable 1 H-pyrrolo [3, 2-c] pyridine inhibitors of mitotic kinase monopolar spindle 1 (MPS1)

S Naud, IM Westwood, A Faisal…

Index: Journal of Medicinal Chemistry, , vol. 56, # 24 p. 10045 - 10065

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Citation Number: 24

Abstract

... Journal of Medicinal Chemistry. ... Kingdom. J. Med. Chem. , 2013, 56 (24), pp 10045–10065. DOI: 10.1021/jm401395s. Publication Date (Web): November 20, 2013. Copyright © 2013 American Chemical Society. *Telephone ...

Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitors via one-pot Sonogashira coupling–TMS-deprotection–CuAAC sequence

[Organic and Biomolecular Chemistry, , vol. 9, # 14 p. 5129 - 5136]

Structure-based design of orally bioavailable 1 H-pyrrolo [3, 2-c] pyridine inhibitors of mitotic kinase monopolar spindle 1 (MPS1)

Abstract

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