Tetrahedron letters

Crystallization-induced asymmetric transformation (CIAT) with simultaneous epimerization at two stereocenters. A short synthesis of conformationally constrained …

A Kolarovič, D Berkeš, P Baran, F Považanec

Index: Kolarovic, Andrej; Berkes, Dusan; Baran, Peter; Povazanec, Frantisek Tetrahedron Letters, 2005 , vol. 46, # 6 p. 975 - 978

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Citation Number: 22

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... CIAT of aza-Michael adducts allows simultaneous build up of two stereocenters. A consequent short and efficient synthesis affords simple access to the both antipodes of various conformationally restricted homophenylalanines. ... Reagents and conditions: (i) 1.1equiv (R)- ...