Tetrahedron Letters

Ortho-amination of lithiated tertiary benzamides. Short route to polysubstituted anthranilamides

JN Reed, V Snieckus

Index: Reed, J. N.; Snieckus, V. Tetrahedron Letters, 1983 , vol. 24, # 36 p. 3795 - 3798

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Citation Number: 36

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Directed lithiation of benzamides (1), phenyloxazoline (4a), methoxymethoxybenzene (4b), and -phenyl carbamate (4c) followed by sequential treatment with TsN 3 and NaBH 4 constitutes a general route to synthetically useful amino aromatics 3 and 5. ... For recent work, see ...