Evaluation and biological properties of reactive ligands for the mapping of the glycine site on the N-methyl-D-aspartate (NMDA) receptor

A Kreimeyer, B Laube, M Sturgess…

Index: Journal of Medicinal Chemistry, , vol. 42, # 21 p. 4394 - 4404

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Citation Number: 35

Abstract

... Journal of Medicinal Chemistry. ... Chemistry. The affinity probes 13a−e and 15a−f, derived from the lead compounds L-701.324 and L-698.532 (Chart 1), were prepared as shown in Scheme 1. The synthesis of ligands ...

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