Substituted furans as inhibitors of the PDE4 enzyme

…, R Rasori, A Robichaud, Y Girard, D Macdonald

Index: Perrier, Helene; Bayly, Christopher; Laliberte, France; Huang, Zheng; Rasori, Roberta; Robichaud, Annette; Girard, Yves; Macdonald, Dwight Bioorganic and Medicinal Chemistry Letters, 1999 , vol. 9, # 3 p. 323 - 326

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Citation Number: 24

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... The synthesis and in vitro activity of a series of substituted furans as a novel structural class of PDE4 inhibitors is described. Comparison of emetic threshold with known PDE4 inhibitors is presented. ... The synthesis and the in vitro activity of a series of substituted furans as a ...

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