Base-Promoted β-C (sp3)–H Functionalization of Enaminones: An Approach to Polysubstituted Pyridines

…, C Kuai, Y Liu, M Wei, G Cheng, X Cui

Index: Shen, Jinhai; Cheng, Guolin; Cui, Xiuling Chemical Communications, 2013 , vol. 49, # 90 p. 10641 - 10643

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Citation Number: 7

Abstract

A convenient “one-pot” base-promoted synthesis of polysubstituted pyridines from 1- arylethylamines and ynones through the direct β-C (sp3)–H functionalization of enaminones under metal-free conditions has been developed. An intermolecular Michael addition