Solid phase synthesis of aryl amines
CA Willoughby, KT Chapman
Index: Willoughby, Christopher A.; Chapman, Kevin T. Tetrahedron Letters, 1996 , vol. 37, # 40 p. 7181 - 7184
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Citation Number: 86
Abstract
A method for the solid phase synthesis of aryl amines is reported. The method involves a palladium mediated coupling reaction between aryl bromides and amines. The products are isolated in high purity and good yields. This method should prove to be a useful tool for constructing combinatorial libraries containing the aryl amine moiety.
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