Multicomponent C??Alkylation Reactions of Aromatic Aldimines with Trialkylboranes Reagents

…, C Muñoz, A Díaz, G Torres, R Suau

Index: Valpuesta, Maria; Munoz, Carmen; Diaz, Amelia; Torres, Gregorio; Suau, Rafael European Journal of Organic Chemistry, 2010 , # 10 p. 1934 - 1942

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Citation Number: 3

Abstract

Abstract The one-pot three-component reaction of an aryl aldehyde, an arylamine, and a trialkylborane in the presence of hydrogen peroxide afforded the alkylated arylamines 1 in good yields via oxidized imine–borane complexes. In addition, the versatility of our procedure has been confirmed by the use of enolizable aldehydes, alkylic amines, and cyclic imines.