N-Acyl glycinates as acyl donors in serine protease-catalyzed kinetic resolution of amines. Improvement of selectivity and reaction rate

M Nechab, L El Blidi, N Vanthuyne…

Index: Organic and Biomolecular Chemistry, , vol. 6, # 21 p. 3917 - 3920

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Citation Number: 15

Abstract

... Chem., 2008, 6, 3917-3920 Show Compounds Show Chemical Terms. ... 5 However, substilisins are generally less reactive, less selective and less stable in an organic medium than ... and ranged between 20 min to 3 h depending on the concentration (entries 4–6). Although the ...

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