Lipase-mediated resolution of inden-1-ol

M Takahashi, R Koike, K Ogasawara

Index: Takahashi; Koike; Ogasawara Chemical and Pharmaceutical Bulletin, 1995 , vol. 43, # 9 p. 1585 - 1587

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Citation Number: 5

Abstract

Optically active inden-l-ol (1) has potential utility as a key starting material for the preparation of HIV-1 protease inhibitors such as L-735,524 and L-754,394.” Synthesis of optically active inden-l-ol (1), however, has been little studied and only one enantiotopical prepara-tion” has

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