Discovery of novel heteroarylazoles that are metabotropic glutamate subtype 5 receptor antagonists with anxiolytic activity
J Roppe, ND Smith, D Huang, L Tehrani…
Index: Journal of Medicinal Chemistry, , vol. 47, # 19 p. 4645 - 4648
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Citation Number: 113
Abstract
... Journal of Medicinal Chemistry. ... The chemical synthesis of the N-linked azole analogues is summarized in Schemes 1−3 (detailed procedures may be found in the Supporting Information). Yields reported are unoptimized. ...
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