Discovery of N-{5-[3-(3-hydroxypiperidin-1-yl)-1, 2, 4-oxadiazol-5-yl]-4-methyl-1, 3-thiazol-2-yl} acetamide (TASP0415914) as an orally potent phosphoinositide 3- …

Y Oka, T Yabuuchi, T Oi, S Kuroda, Y Fujii…

Index: Bioorganic and Medicinal Chemistry, , vol. 21, # 24 p. 7578 - 7583

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Abstract

... Bioorganic & Medicinal Chemistry. ... a Medicinal Chemistry Laboratories, Taisho ... c Pharmacokinetics and Metabolism Drug Safety and Pharmacokinetics Laboratories, Taisho Pharmaceutical Co., Ltd, 1-403, Yoshino-Cho, Kita-Ku, Saitama-Shi, Saitama 331-9530, Japan. ...

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