Synthesis of Symmetric Diester??Functionalised Tröger's Base Analogues

MDH Bhuiyan, KX Zhu, P Jensen…

Index: Bhuiyan, M. Delower H.; Zhu, Kai-Xian; Jensen, Paul; Try, Andrew C. European Journal of Organic Chemistry, 2010 , # 24 p. 4662 - 4670

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Citation Number: 8

Abstract

Abstract The yields of ester-functionalised Tröger's base analogues are dramatically improved by incorporating an electron-donating group on the aromatic ring and/or enhancing solubility of the aniline unit. In addition to 2, 8-diester compounds, 1, 7-, 3, 9-and 4, 10-diester-functionalised Tröger's base analogues have been prepared for the first time.

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