Tetrahedron letters

Enantioselective one-pot synthesis of β-lactams from achiral 2-pyridylthioesters and aromatic imines

R Annunziata, M Benaglia, M Cinquini, F Cozzi

Index: Annunziata, Rita; Benaglia, Maurizio; Cinquini, Mauro; Cozzi, Franco Tetrahedron Letters, 1995 , vol. 36, # 4 p. 613 - 616

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Citation Number: 17

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... The enolates derived from 2-pyridylthioesters by reaction with BCl 3 ·SMe 2 and enantiomerically pure aminoalcohols react with aromatic imines in an enantioselective fashion (ee up to 78%) to afford β-lactams in a convenient one-pot procedure. ... The enolates derived from 2- ...