Some Derivatives of Benzoyl and Furoyl Isothiocyanates and their Use in Synthesizing Heterocyclic Compounds1

IB Douglass, FB Dains

Index: Douglass; Dains Journal of the American Chemical Society, 1934 , vol. 56, p. 719

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Citation Number: 178

Abstract

Benzoyl isothiocyanate readily combines with arylaminoethanols, phenylaminopropanol, phenylaminoacetic acid, or anthranilic acid. Dehydration of the resulting thioureas yields thiazolidines, a thiazane, a 2-thioimidazolone, or a quinazoline derivative as the case may be. Desulfurization of the acylethanolthioureas results in forming oxazolidines. Some thirty acyl isothiocyanates are described in the literature but none is derived from a heterocyclic ...