1, 5-Substituted nipecotic amides: selective PDE8 inhibitors displaying diastereomer-dependent microsomal stability

MP DeNinno, SW Wright, MS Visser, JB Etienne…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 10 p. 3095 - 3098

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Citation Number: 20

Abstract

... Bioorganic & Medicinal Chemistry Letters. Volume 21, Issue 10, 15 May 2011, Pages 3095–3098. Cover image Cover image. 1,5-Substituted nipecotic amides: Selective PDE8 inhibitors displaying diastereomer-dependent microsomal stability. ...

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