Novel 3-azaindolyl-4-arylmaleimides exhibiting potent antiangiogenic efficacy, protein kinase inhibition, and antiproliferative activity

…, T Stauder, JP Kramb, S Plutizki, T Kindler…

Index: Cash, Michael T.; Schreiner, Peter R.; Phillips, Robert S. Organic and Biomolecular Chemistry, 2005 , vol. 3, # 20 p. 3701 - 3706

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Citation Number: 16

Abstract

... Journal of Medicinal Chemistry. ... respectively, using vinylmagnesium bromide and catalytic hydrogenation.(9) In the case of 4-azaindole, procedures by Cash et al ... esters (10d, 11a–c) and arylacetamide derivatives (12a–c) in the presence of potassium tert-butoxide ( t BuOK) and ...

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