Discovery and optimisation of a selective non-steroidal glucocorticoid receptor antagonist

AR Brown, M Bosies, H Cameron, J Clark…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 1 p. 137 - 140

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Citation Number: 11

Abstract

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. Volume 21, Issue 1, 1 January 2011, Pages 137–140. ... Compd, R 1, R 2, R 3, Stereo chemistry, C log P, GR 10 pEC 50, PR 10 pEC 50, Binding selectivity PR/GR. ...

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