A novel, potent, and selective 5-HT7 antagonist:(R)-3-(2-(2-(4-methylpiperidin-1-yl)-ethyl) pyrrolidine-1-sulfonyl) phenol (SB-269970)

…, DN Middlemiss, SK Rahman, DV Saunders…

Index: Lovell, Peter J.; Bromidge, Steven M.; Dabbs, Steven; Duckworth, D. Malcolm; Forbes, Ian T.; Jennings, Andrew J.; King, Frank D.; Middlemiss, Derek N.; Rahman, Shirley K.; Saunders, Damian V.; Collin, Lissa L.; Hagan, Jim J.; Riley, Graham J.; Thomas, David R. Journal of Medicinal Chemistry, 2000 , vol. 43, # 3 p. 342 - 345

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Citation Number: 234

Abstract

... SB-269970). Auteur(s) / Author(s). LOVELL PJ (1) ; BROMIDGE SM (1) ; DABBS S. (1) ; DUCKWORTH DM (1) ; FORBES IT (1) ; JENNINGS AJ (1) ; KING FD (1) ; MIDDLEMISS DN (1) ; RAHMAN SK (1) ; SAUNDERS DV (1) ; COLLIN LL (1) ; HAGAN JJ (1) ; RILEY GJ (1) ; THOMAS DR (1) ; Affiliation(s) du ou des auteurs / Author(s) Affiliation(s). (1) SmithKline ...

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