Transition metal catalyzed synthesis of 5-azaindoles
L Xu, IR Lewis, SK Davidsen, JB Summers
Index: Xu, Lianhong; Lewis, Iestyn R.; Davidsen, Steven K.; Summers, James B. Tetrahedron Letters, 1998 , vol. 39, # 29 p. 5159 - 5162
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Citation Number: 89
Abstract
In an effort to develop synthetic procedures for the preparation of 2-substituted 5-azaindoles, the synthesis and cyclization reactions of acetylenic aminopyridines was explored. A novel method for the synthesis of 2-substituted 5-azaindoles via a transition metal catalyzed reaction is described.
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