Microwave??Assisted [3+ 2] Cycloaddition and Suzuki–Miyaura Cross??Coupling for a Concise Access to Polyaromatic Scaffolds
D Hedou, E Deau, C Dubouilh??Benard…
Index: Hedou, Damien; Deau, Emmanuel; Dubouilh-Benard, Carole; Sanselme, Morgane; Martinet, Anthony; Chosson, Elizabeth; Levacher, Vincent; Besson, Thierry European Journal of Organic Chemistry, 2013 , # 33 p. 7533 - 7545
Full Text: HTML
Citation Number: 4
Abstract
Abstract Novel 3-(prop-2-ynyl) pyrido [2, 3-d] pyrimidin-4 (3H)-ones and 3-(prop-2-ynyl) quinazolin-4 (3H)-ones have been synthesized in a high-yielding microwave-assisted one- pot procedure. The one-pot sequence was conveniently extended to the synthesis of commercially unavailable 6-bromo-N 3-propargylpyrido [2, 3-d] pyrimidinone by a regiocontrolled bromination with NBS. The synthetic scaffolds were successfully converted ...
Related Articles:
[Iranpoor, Nasser; Firouzabadi, Habib; Akhlaghinia, Batool; Nowrouzi, Najmeh Tetrahedron Letters, 2004 , vol. 45, # 16 p. 3291 - 3294]
Synthesis and phytotoxic activity of 1, 2, 3-triazole derivatives
[Borgati, Thiago F.; Alves, Rosemeire B.; Teixeira, Robson R.; De Freitas, Rossimiriam P.; Perdigao, Thays G.; Da Silva, Silma F.; Dos Santos, Aline Aparecida; De Jesus O. Bastidas, Alberto Journal of the Brazilian Chemical Society, 2013 , vol. 24, # 6 p. 953 - 961]
[Pramanik, Suman; Ghorai, Prasanta Organic Letters, 2014 , vol. 16, # 8 p. 2104 - 2107]
[Buckley, Neil; Oppenheimer, Norman J. Journal of Organic Chemistry, 1996 , vol. 61, # 21 p. 7360 - 7372]