Tetrahedron

Convenient access to substituted acridines by a Buchwald–Hartwig amination

R Csuk, A Barthel, C Raschke

Index: Csuk, Rene; Barthel, Alexander; Raschke, Christian Tetrahedron, 2004 , vol. 60, # 27 p. 5737 - 5750

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Citation Number: 43

Abstract

A convenient, high yield procedure for the synthesis of anthranilic acids carrying a variety of different substituents as well as their straightforward transformation into the corresponding 9- chloroacridines could be established by using modified Buchwald–Hartwig amination conditions.