First Suzuki–Miyaura type cross-coupling of ortho-azidobromobenzene with arylboronic acids and its application to the synthesis of fused aromatic indole-heterocycles
M Pudlo, D Csányi, F Moreau, G Hajós, Z Riedl, J Sapi
Index: Pudlo, Marc; Csanyi, Dorottya; Moreau, Fabien; Hajos, Gyoergy; Riedl, Zsuzsanna; Sapi, Janos Tetrahedron, 2007 , vol. 63, # 41 p. 10320 - 10329
Full Text: HTML
Citation Number: 38
Abstract
A short synthesis of some fused indole-heterocycles has been achieved via Pd-catalyzed cross-coupling reactions between azido-2-bromobenzene and arylboronic acids and subsequent thermally induced nitrene insertion. Additionally, 4-amino-α-carboline, a versatile intermediate toward grossularine analogs has also been prepared by Suzuki– Miyaura cross-coupling of 4-pivaloylaminopyridine-3-boronic acid with 2-bromoaniline, ...
Related Articles:
General Copper??Catalyzed Transformations of Functional Groups from Arylboronic Acids in Water
[Yang, Haijun; Li, Yong; Jiang, Min; Wang, Junmei; Fu, Hua Chemistry - A European Journal, 2011 , vol. 17, # 20 p. 5652 - 5660]
The Physical Properties of Some Triazo Compounds. I. Molar Refractions and Parachors1
[Spauschus; Scott Journal of the American Chemical Society, 1951 , vol. 73, p. 208]
Click chemistry inspired facile synthesis and bioevaluation of novel triazolyl analogs of Ludartin
[Lone, Shabir H.; Bhat, Khursheed A.; Majeed, Rabiya; Hamid, Abid; Khuroo, Mohd A. Bioorganic and Medicinal Chemistry Letters, 2014 , vol. 24, # 4 p. 1047 - 1051]