Diarylthiazole: an antimycobacterial scaffold potentially targeting PrrB-PrrA two-component system
E Bellale, M Naik, A Ambady, A Narayan…
Index: DAIICHI PHARMACEUTICAL CO., LTD Patent: US2003/92720 A1, 2003 ;
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Citation Number: 10
Abstract
... Interestingly, both electron-withdrawing and electron-donating groups were active. Furthermore, substituents at ortho, meta, and para positions were found to be equipotent from the limited set of electron-withdrawing and electron-donating groups explored (Table 2, 13–21). ...
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