Tetrahedron

Brief syntheses of (+)-blastmycinone and related γ-lactones from an asymmetrically dihydroxylated carboxylic ester

T Berkenbusch, R Brückner

Index: Berkenbusch, Thilo; Brueckner, Reinhard Tetrahedron, 1998 , vol. 54, # 38 p. 11461 - 11470

Full Text: HTML

Citation Number: 41

Abstract

A method for synthesizing optically active trans, trans-configurated α, β, γ-substituted γ- lactones is presented. Asymmetric hydroxylation of ester 8 with AD mix α (AD mix β) and subsequent dehydration provided butenolide S-6 (R-6). Conjugate addition of Li2 (Me2PhSi) 2Cu (CN) to S-6 followed by alkylation of the resulting enolate led to the stereopure silyllactones 9–11. They furnished the title compounds after oxidative removal ...

Related Articles:

Improved syntheses of high hole mobility phthalocyanines: A case of steric assistance in the cyclo-oligomerisation of phthalonitriles

[Tate, Daniel J.; Anemian, Remi; Bushby, Richard J.; Nanan, Suwat; Warriner, Stuart L.; Whitaker, Benjamin J. Beilstein Journal of Organic Chemistry, 2012 , vol. 8, p. 120 - 128]

Über Alken??(1)??ine??(4)

[Justus Liebigs Annalen der Chemie, , vol. 658, p. 6 - 20]

Volatile methyl esters of medium chain length from the bacterium Chitinophaga Fx7914

[Nawrath, Thorben; Gerth, Klaus; Mueller, Rolf; Schulz, Stefan Chemistry and Biodiversity, 2010 , vol. 7, # 9 p. 2228 - 2253]

Wax composition of Sargassum fulvellum

[Miyazawa, Mitsuo; Uematsu, Tosihisa; Kameoka, Hiromu Phytochemistry (Elsevier), 1982 , vol. 21, # 7 p. 1788 - 1791]

Synthesis and pharmacology of the isomeric methylheptyl-Δ 8-tetrahydrocannabinols

[Bioorganic and Medicinal Chemistry, , vol. 6, # 12 p. 2383 - 2396]

More Articles...