Synthesis of some 2-aryl-1, 2, 4-triazolo [1, 5-c][1, 3] benzoxazin-5-ones as tools to define the essential pharmacophoric descriptors of a benzodiazepine receptor …

D Catarzi, L Cecchi, V Colotta…

Index: Journal of Medicinal Chemistry, , vol. 38, # 12 p. 2196 - 2201

Full Text: HTML

Citation Number: 20

Abstract

... 0 1995 American Chemical Society Page 2. 2-Aryl-l,2,4-triazolo[l,5-cl[l,3]benzoxazin-5-ones Scheme 2a Journal of Medicinal Chemistry, 1995, Vol. 38, No. 12 2197 ._. . 23 24: K = tI 25: R = C1 a (a) Et3N/CHzClz; (b) heating over their melting points. ...