The Synthesis of a New Class of Potential Inhibitors for Glycoside Hydrolases†
RV Stick, KA Stubbs
Index: Stick, Robert V.; Stubbs, Keith A. Journal of Carbohydrate Chemistry, 2005 , vol. 24, # 4-6 p. 529 - 547
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Citation Number: 9
Abstract
Some attempts toward the synthesis of novel inhibitors of glycosyl transferases are described. More successfully, the synthesis of an activated cyclopropacyclohexene and an amide and an amine of a cyclopropa??fused pyranose are described. None of these three novel compounds proved to be a significant inhibitor of a retaining α??glucosidase from barley.† This paper is dedicated to the memory of Jacques H. van Boom.
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