Tetrahedron letters

Nitrogen Alkylation of schiff bases and amidines as a route to N-alkyl amino acids

MJ O'Donnell, WA Bruder, BW Daugherty, D Liu…

Index: O'Donnell, Martin J.; Bruder, William A.; Daugherty, Byron W.; Liu, Deshan; Wojciechowski, Krzisztof Tetrahedron Letters, 1984 , vol. 25, # 34 p. 3651 - 3654

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Citation Number: 28

Abstract

This document does not have an outline. ... JavaScript is disabled on your browser. Please enable JavaScript to use all the features on this page. ... Author links open the overlay panel. Numbers correspond to the affiliation list which can be exposed by using the show more link. ... Schiff base and amidine ester 3 are alkylated and then hydrolyzed to yield N-alkyl amino acids 4 in 41–75% yield with high to complete retention of optical activity.

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