Heterocycles

New synthetic approach to 1-azabicyclo [xy 0] alkane skeletons from β-enamino diesters derived from Meldrum's acid

…, JP Célérier, G Haviari, G Lhommet, H Dhimane…

Index: Haddad, Mansour; Celerier, Jean Pierre; Haviari, Gjergj; Lhommet, Gerard; Dhimane, Hamid; at al. Heterocycles, 1990 , vol. 31, # 7 p. 1251 - 1260

Full Text: HTML

Citation Number: 12

Abstract

Résumé/Abstract Two complementary methods for the synthesis of title compounds, namely, monodecarboxylating transesterification of β-enamino esters (I) followed by intramolecular cyclization, and direct cyclization of I under flash vacuum thermolysis conditions, have been elaborated. Azabicyclic compounds were stereospecifically converted to bicyclic β-amino alcohols by means of stereocontrolled carbon-carbon double bond catalytic ...

Related Articles:

β-Enaminoesters bicycliques: Synthese et reduction stereospecifiques. Acces a l'isoretronecanol, la trachelanthamidine, la lupinine et l'epilupinine

[Celerier, J. P.; Haddad, M.; Saliou, C.; Lhommet, G. Tetrahedron, 1989 , vol. 45, # 19 p. 6161 - 6170]

More Articles...