Diazinones as P2 replacements for pyrazole-based cathepsin S inhibitors

MK Ameriks, SD Bembenek, MT Burdett…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 14 p. 4060 - 4064

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Abstract

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. Volume 20, Issue 14, 15 July 2010, Pages 4060–4064. Cover image Cover image. ... In this letter, we describe how a low-affinity pyridazinone fragment 4 (Fig. ...

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