Rapid synthesis of 2, 5??disubtituted 1, 3, 4??thiadiazoles under microwave irradiation
M Lebrini, F Bentiss, M Lagrenée
Index: Lebrini, Mounim; Bentiss, Fouad; Lagrenee, Michel Journal of Heterocyclic Chemistry, 2005 , vol. 42, # 5 p. 991 - 994
Full Text: HTML
Citation Number: 48
Abstract
Abstract The one pot, three-components condensation of aromatic aldehydes, hydrazine and sulfur in ethanol under microwave irradiation provided symmetrically 3, 5-disubstituted 1, 3, 4-thiadiazoles in high yields and good purity. This reaction must be conducted under pressure of hydrogen sulfide produced in-situ. The structure of the compounds was confirmed by 1 H, 13 C NMR, MS and elemental analysis.
Related Articles:
[Klingele, Julia; Kaase, Dominic; Klingele, Marco H.; Lach, Jochen Dalton Transactions, 2012 , vol. 41, # 4 p. 1397 - 1406]
[Geldard,J.F.; Lions,F. Journal of Organic Chemistry, 1965 , vol. 30, p. 318 - 319]