Tetrahedron

Novel series of 8H-quinazolino [4, 3-b] quinazolin-8-ones via two Niementowski condensations

FR Alexandre, A Berecibar, R Wrigglesworth, T Besson

Index: Alexandre, Francois-Rene; Berecibar, Amaya; Wrigglesworth, Roger; Besson, Thierry Tetrahedron, 2003 , vol. 59, # 9 p. 1413 - 1419

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Citation Number: 82

Abstract

Efficient microwave-assisted multi-step synthesis of 8H-quinazolino [4, 3-b] quinazolin-8-one was investigated. The synthesis involved two Niementowski condensations from anthranilic acids. Homogeneous or heterogeneous conditions were studied with the aim to develop convenient syntheses of the desired compounds.

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