Tetrahedron letters

Selective alkylation of a 6, 7-dihydroxyquinazoline

CS Harris, LF Hennequin, JG Kettle, OA Willerval

Index: Harris, Craig S.; Hennequin, Laurent F.; Kettle, Jason G.; Willerval, Olivier A. Tetrahedron Letters, 2005 , vol. 46, # 45 p. 7715 - 7719

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Citation Number: 17

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... A convenient 3-step multi-parallel process for the preparation of 4-(3-chloro-2-fluoroanilino)-6,7-bisalkoxyquinazolines is highlighted. ... Examples of anilinoquinazolines in clinical development. Examples of anilinoquinazolines in clinical development. ... In our recent efforts to explore variation at positions C-6 and ...

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